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Drug Interaction Information in Human Prescription Drug and Biological Product Labeling

DraftCenter for Drug Evaluation and Research10/21/2024

Description

This guidance is intended to assist applicants of human prescription drug and biological products in determining the appropriate placement and content of drug interaction (DI) information in labeling as described in the regulations for the content and format of labeling for human prescription drug and biological products. The purpose of this guidance is to provide recommendations to help ensure that appropriate DI information is consistently placed in the proper sections and subsections within labeling so that the information is clear and accessible to health care practitioners (HCPs) and includes content that guides the safe and effective use of the drug.

Scope & Applicability

Product Classes

4
Human Prescription Drug

guidance applies to drugs regulated under section 505

Biological Product

Regulated under section 351(i) of the PHS Act; Virus, therapeutic serum, toxin, vaccine, or protein applicable to prevention or treatment; Alternative regulation category for products meeting device definition

Therapeutic Proteins

Proteins that reduce proinflammatory cytokines and affect CYP enzyme expression

Tyrosine Kinase Inhibitors

Example of a drug class known for specific interactions

Stakeholders

5
Health Care Practitioners

ensure information is clear and accessible to HCPs

Applicant

Entity submitting development data and knowledge; Entity performing the work process for change

HCPs

Healthcare professionals who reference labeling and public resources

Applicants

Entities submitting supplements to BLAs

Health Care Professionals

The target audience for labeling information.

Regulatory Context

Attributes

3
Clinically significant

Threshold for including drug interaction information in labeling.

Cmax

Cmax may be more informative for safety

AUC

AUC or Cmin may correlate with efficacy

Identified Hazards

Hazards

3
Risk of bleeding

Example of a specific clinical effect from a DI

Drug resistance

Potential safety issue from drug interactions

Treatment failure

Clinically significant outcome of a drug interaction

Related CFR Sections (2)

See Also (8)

Drug Interaction Information in Human Prescription Drug and Biological Product Labeling | Guideline Explorer | BioRegHub