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Hypertension: Developing Fixed-Dose Combination Drugs for Treatment

FinalCenter for Drug Evaluation and Research11/07/2018
Pharmacokinetics

Description

The Food and Drug Administration (FDA or Agency) is announcing the availability of a final guidance for industry entitled “Hypertension: Developing Fixed-Combination Drug Products for Treatment.” The purpose of this guidance is to assist sponsors in the clinical development of fixed-combination drug products for the treatment of hypertension. The guidance focuses on development of two-drug combinations of previously approved drug products. This guidance incorporates the comments received for and finalizes the draft guidance for industry entitled “Hypertension: Developing Fixed-Dose Combination Drugs for Treatment” issued on January 26, 2018.

Key Topics

Terms and concepts identified from this document

Scope & Applicability

Product Classes

2
Fixed-Dose Combination Drugs

Developing fixed-dose combination drugs for hypertension treatment

Fixed-Combination Drug Product

Two or more active ingredients combined at a fixed dosage

Stakeholders

1
Sponsor

Entity responsible for submitting applications under section 524B

Regulatory Context

Regulatory Activities

1
Phase 3 Trial

Sponsors should conduct two randomized, double-blind, controlled trials.

Document Types

1
Labeling

Cybersecurity information should be included in device labeling

Attributes

1
Blood pressure

measured in millimeters of mercury (mmHg)

Technical Details

Substances

4
Beta blocker

drug product with distinct mechanism of action

Angiotensin-receptor blocker

drug product with distinct mechanism of action

Angiotensin-converting enzyme inhibitor

drug product with distinct mechanism of action

Diuretic

drug product with distinct mechanism of action

Testing Methods

1
Factorial Study

using multiple doses of each component to show contribution; Comparing A plus B to A and to B at their highest approved doses

Clinical Concepts

6
Diastolic blood pressure

Significant effects are observed on both systolic and diastolic blood pressures

Systolic blood pressure

Significant effects are observed on both systolic and diastolic blood pressures

Blood pressure effect

Showing that each component contributes to the blood pressure effect

Coronary artery disease

Closely related population to heart failure

Stroke

correlated with female sex in VAD study

Hypertension

comorbidity associated with obesity; Common weight-related comorbidity; Weight-related comorbidity

Standards & References

External Standards

1
Treatment guidelines

Sponsors should consult contemporary treatment guidelines

Related CFR Sections (1)

Related MFDS Guidelines

Korean regulatory guidelines covering similar topics

See Also (8)

Hypertension: Developing Fixed-Dose Combination Drugs for Treatment | Guideline Explorer | BioRegHub